SCHEMBL9723264

SCHEMBL9723264

CCCCCCCc1ccc(C#N)c(F)c1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYR P14679 3/20 0.44
TSHR P16473 2/20 0.44
TP53 P04637 2/20 0.44
CYP3A4 P08684 2/20 0.44
MEN1 O00255 1/20 0.44
ALOX5 P09917 1/20 0.44
MAPT P10636 1/20 0.44
ALOX15 P16050 1/20 0.44
HTT P42858 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HSD17B10 Q99714 2/20 0.41
ALDH1A1 P00352 2/20 0.38
LIPG Q9Y5X9 1/20 0.38
HPGD P15428 1/20 0.38
AR P10275 2/20 0.35
ESR1 P03372 2/20 0.33
ADRA2A P08913 2/20 0.33
ADORA3 P0DMS8 2/20 0.33
TACR2 P21452 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9723171 0.98 TYR (0.41) TYRTSHRTP53CYP3A4MEN1
SCHEMBL9723274 0.86 AR (0.40) TDP1AR
SCHEMBL9710392 0.83 TYR (0.44) TYRTSHRTP53CYP3A4MEN1
SCHEMBL9710325 0.83 TYR (0.44) TYRTSHRTP53CYP3A4MEN1
SCHEMBL10520219 0.83 TYR (0.44) TYRTSHRTP53CYP3A4MEN1
SCHEMBL9710309 0.83 TYR (0.44) TYRTSHRTP53CYP3A4MEN1
SCHEMBL9447304 0.82 HTR2A (0.36) TSHRCYP3A4MAPTHSD17B10ALDH1A1
SCHEMBL9447300 0.82 HTR2A (0.36) TSHRCYP3A4MAPTHSD17B10ALDH1A1
SCHEMBL9447155 0.82 HTR2A (0.36) TSHRCYP3A4MAPTHSD17B10ALDH1A1
SCHEMBL9447150 0.82 HTR2A (0.36) TSHRCYP3A4MAPTHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5087764-A Deprotonation of a 1-substituted-2,3-difluorobenzene using an organometallic compound and reacting the reaction product with an electrophile Merck Patent Gesellschaft mit beschrankter Hafung (DE) 1992-02-11 US disclosed
CN-1037327-A Preparation 2, the method for 3-phenyl-difluoride class MERCK PATENT GMBH (DE) 1989-11-22 CN disclosed