SCHEMBL9726173

SCHEMBL9726173

O=[N+]([O-])c1cc(Cl)ccc1CC(O)=S

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.50
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
MAPK1 P28482 3/20 0.47
TSHR P16473 1/20 0.47
VCAM1 P19320 1/20 0.45
PDE7A Q13946 2/20 0.44
PDE7B Q9NP56 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
CYP3A4 P08684 2/20 0.44
HPGD P15428 2/20 0.44
CYP2C19 P33261 2/20 0.44
ACLY P53396 1/20 0.44
KIF18A Q8NI77 1/20 0.43
APP P05067 1/20 0.43
PDE4B Q07343 1/20 0.42
PDE4D Q08499 1/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9726177 1.00 CYP1A2 (0.50) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL10511030 0.87 TSHR (0.51) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL10511033 0.87 TSHR (0.51) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL442788 0.85 CYP1A2 (0.69) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL9452749 0.85 CYP1A2 (0.69) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL7827901 0.84 CYP1A2 (0.54) CYP1A2NPC1RAB9AMAPK1TSHR
Hydrochloric Acid SCHEMBL11329805 0.84 CYP1A2 (0.67) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL11329796 0.82 NPC1 (0.52) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL29836060 0.81 MAPK1 (0.52) CYP1A2NPC1RAB9AMAPK1TSHR
SCHEMBL535457 0.81 MAPK1 (0.52) CYP1A2NPC1RAB9AMAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5141935-A Dihydrobenz thiazine derivative and microorganism control agent UBE INDUSTRIES, LTD. (JP) 1992-08-25 US disclosed
EP-0162776-B1 HETEROCYCLIC DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS USEFUL AS ALDOSE REDUCTASE INHIBITORS CONTAINING THEM LABORATOIRES UPSA (FR) 1989-04-19 EP disclosed
EP-0162776-A2 Heterocyclic derivatives, process for their preparation and medicaments useful as aldose reductase inhibitors containing them LABORATOIRES UPSA (FR) 1985-11-27 EP disclosed