SCHEMBL9728693

SCHEMBL9728693

NC(=O)c1ccccc1-c1ncc2ccccc2n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.49
CSNK1A1 P48729 2/20 0.48
DYRK1B Q9Y463 2/20 0.48
TYRO3 Q06418 1/20 0.48
IKBKB O14920 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
MAPK1 P28482 1/20 0.47
CYP2C19 P33261 1/20 0.47
BCAT2 O15382 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
GRM5 P41594 1/20 0.44
PARP1 P09874 4/20 0.41
NUDT1 P36639 1/20 0.40
PLK4 O00444 1/20 0.40
CHEK1 O14757 1/20 0.40
AURKA O14965 1/20 0.40
DAPK3 O43293 1/20 0.40
MAP4K4 O95819 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30306357 1.00 CYP1A2 (0.49) CYP1A2CSNK1A1DYRK1BTYRO3IKBKB
SCHEMBL12276902 0.88 IKBKB (0.47) CYP1A2CSNK1A1DYRK1BTYRO3IKBKB
SCHEMBL30670415 0.86 CYP1A2 (0.50) CYP1A2NPC1RAB9AKDM4EALDH1A1
SCHEMBL27029796 0.86 CYP1A2 (0.50) CYP1A2NPC1RAB9AKDM4EALDH1A1
SCHEMBL27600087 0.83 IKBKB (0.44) CYP1A2IKBKBCYP3A4CYP2D6MAPK1
SCHEMBL27029841 0.81 KMT2A (0.51) CYP1A2KDM4EALDH1A1
SCHEMBL12276898 0.80 IKBKB (0.47) CYP1A2CSNK1A1DYRK1BIKBKBMAPK1
SCHEMBL31679004 0.77 IKBKB (0.47) CYP1A2IKBKBRAB9APARP1ROCK2
SCHEMBL19143038 0.75 CYP1A2 (0.56) CYP1A2CYP3A4CYP2D6MAPK1CYP2C19
SCHEMBL31116679 0.75 CYP1A2 (0.56) CYP1A2CYP3A4CYP2D6MAPK1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084457-A Cognition activators and nervous system disorders AMERICAN CYANAMID COMPANY (US) 1992-01-28 US disclosed