SCHEMBL9730453

SCHEMBL9730453

CN(C)c1ccccc1CC(=O)N1CC2C(=O)CCC(c3ccccc3F)(c3ccccc3F)C2C1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.57
MEN1 O00255 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
FNTA P49354 3/20 0.38
FNTB P49356 3/20 0.38
OPRD1 P41143 4/20 0.36
OPRK1 P41145 4/20 0.36
RORC P51449 1/20 0.32
OPRM1 P35372 3/20 0.31
BRD4 O60885 1/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9730940 0.99 TACR1 (0.56) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9373109 0.87 TACR1 (0.68) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9272085 0.87 TACR1 (0.68) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9730542 0.85 TACR1 (0.59) TACR1MEN1CYP3A4MAPTTSHR
Hydrochloric Acid SCHEMBL9730405 0.84 TACR1 (0.58) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9730357 0.81 TACR1 (0.54) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9729135 0.80 TACR1 (0.55) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9729686 0.79 TACR1 (0.58) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9730090 0.77 TACR1 (0.56) TACR1MEN1CYP3A4MAPTTSHR
SCHEMBL9729277 0.77 TACR1 (0.36) TACR1DDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112988-A ISOINDOLONE DERIVATIVES RHONE-POULENC SANTE (FR) 1992-05-12 US disclosed