SCHEMBL9736710

SCHEMBL9736710

CN(Cc1ccc2ccccc2n1)C[C@@H](O)COc1ccc(NS(C)(=O)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.54
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
MAPK1 P28482 1/20 0.54
CYP2C19 P33261 1/20 0.54
ADRB2 P07550 1/20 0.47
ADRB1 P08588 1/20 0.47
ADRB3 P13945 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9737861 1.00 KCNH2 (0.54) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9732998 1.00 KCNH2 (0.54) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9737586 0.90 KCNH2 (0.55) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9737387 0.89 KCNH2 (0.52) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9736929 0.88 KCNH2 (0.54) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9736963 0.88 KCNH2 (0.54) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9738723 0.87 KCNH2 (0.57) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9738000 0.87 KCNH2 (0.53) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9737146 0.87 KCNH2 (0.53) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9736514 0.87 KCNH2 (0.53) KCNH2CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084463-A Cardiovascular disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-01-28 US claimed
US-5084463-A Cardiovascular disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-01-28 US disclosed