SCHEMBL9737357

SCHEMBL9737357

Cc1ccc([C@H]2Sc3cc(C)ccc3N(CCN(C)C)C(=O)[C@H]2O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1S Q13698 8/20 0.56
CYP3A4 P08684 3/20 0.46
TSHR P16473 2/20 0.46
ABCB11 O95342 2/20 0.46
LMNA P02545 2/20 0.46
KCNH2 Q12809 2/20 0.46
CACNA1C Q13936 2/20 0.46
SLC22A1 O15245 1/20 0.46
CACNA1F O60840 1/20 0.46
ABCB1 P08183 1/20 0.46
HRH2 P25021 1/20 0.46
ADRA1A P35348 1/20 0.46
SCN1A P35498 1/20 0.46
SCN4A P35499 1/20 0.46
HTT P42858 1/20 0.46
SCN7A Q01118 1/20 0.46
CACNA1D Q01668 1/20 0.46
PLAUR Q03405 1/20 0.46
SCN5A Q14524 1/20 0.46
SCN9A Q15858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9737373 1.00 CACNA1S (0.56) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL7442511 1.00 CACNA1S (0.56) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10640099 0.92 CACNA1S (0.69) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10640105 0.92 CACNA1S (0.69) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10640113 0.92 CACNA1S (0.69) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10636560 0.90 CACNA1S (0.72) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10636573 0.90 CACNA1S (0.72) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10969664 0.90 CACNA1S (0.72) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL12557671 0.89 CACNA1S (0.61) CACNA1SCYP3A4TSHRABCB11LMNA
SCHEMBL10541270 0.89 CACNA1S (0.61) CACNA1SCYP3A4TSHRABCB11LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134139-A Antiarrhythmia agents, blood metal antagonist, hypotensive agents or vasodilator agents TANABE SEIYAKU CO., LTD. (JP) 1992-07-28 US disclosed