SCHEMBL9739359

SCHEMBL9739359

COc1ccc(CCN2CCCC2C(C)N2CCc3cc(OC)c(OC)cc3CC2=O)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 2/20 0.50
MAPT P10636 1/20 0.50
CYP3A4 P08684 1/20 0.49
ALOX15 P16050 1/20 0.49
DHCR7 Q9UBM7 1/20 0.43
ALDH1A1 P00352 6/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
GAA P10253 2/20 0.43
POLB P06746 1/20 0.42
LMNA P02545 3/20 0.41
HTT P42858 2/20 0.41
MAPK1 P28482 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP2D6 P10635 1/20 0.40
HSP90AA1 P07900 1/20 0.39
PAX8 Q06710 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740219 0.97 HCN4 (0.49) HCN4MAPTCYP3A4ALOX15DHCR7
SCHEMBL9740525 0.96 HCN4 (0.49) HCN4MAPTCYP3A4ALOX15DHCR7
Hydrochloric Acid SCHEMBL9740037 0.96 CYP3A4 (0.50) HCN4MAPTCYP3A4ALOX15DHCR7
SCHEMBL9741585 0.89 POLB (0.44) HCN4MAPTCYP3A4ALOX15ALDH1A1
SCHEMBL9739319 0.89 SMN1; SMN2 (0.42) HCN4MAPTCYP3A4ALOX15ALDH1A1
SCHEMBL9740418 0.89 ABCB1 (0.46) HCN4MAPTCYP3A4ALOX15ALDH1A1
Hydrochloric Acid SCHEMBL9739564 0.88 CYP3A4 (0.41) HCN4MAPTCYP3A4ALOX15ALDH1A1
Hydrochloric Acid SCHEMBL9740153 0.88 ABCB1 (0.45) HCN4MAPTCYP3A4ALOX15ALDH1A1
SCHEMBL9739180 0.88 SMN1; SMN2 (0.43) HCN4MAPTCYP3A4ALOX15ALDH1A1
SCHEMBL9739027 0.88 SMN1; SMN2 (0.42) HCN4MAPTCYP3A4ALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed