SCHEMBL9740225

SCHEMBL9740225

CC1COc2c(N3CCC(N)C3)c(F)c(N)c3c(=O)c(C(=O)O)cn1c23

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.56
POLB P06746 3/20 0.52
CACNA1F O60840 1/20 0.52
MAPK1 P28482 1/20 0.52
CACNA1D Q01668 1/20 0.52
KCNH2 Q12809 1/20 0.52
CACNA1S Q13698 1/20 0.52
CACNA1C Q13936 1/20 0.52
AADAT Q8N5Z0 2/20 0.52
KDM4E B2RXH2 4/20 0.51
ALDH1A1 P00352 3/20 0.51
HPGD P15428 2/20 0.51
HSD17B10 Q99714 2/20 0.51
ALB P02768 1/20 0.51
HRH3 Q9Y5N1 1/20 0.51
TOP2A P11388 3/20 0.50
TOP2B Q02880 2/20 0.50
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8684414 0.99 GSK3B (0.55) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL9740204 0.89 GSK3B (0.54) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL10684313 0.86 KDM4E (0.68) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL29391130 0.86 KDM4E (0.68) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL9740963 0.86 GSK3B (0.53) GSK3BPOLBCACNA1FMAPK1CACNA1D
Hydrochloric Acid SCHEMBL29409478 0.85 KDM4E (0.67) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL9739915 0.85 GSK3B (0.52) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL10701430 0.84 GSK3B (0.54) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL9742236 0.84 GSK3B (0.52) GSK3BPOLBCACNA1FMAPK1CACNA1D
SCHEMBL9740992 0.84 GSK3B (0.54) GSK3BPOLBCACNA1FMAPK1CACNA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5097032-A Quinoline- and naphthyridine carboxylic acids, salts WARNER-LAMBERT COMPANY (US) 1992-03-17 US disclosed
EP-0172651-B1 Substituted-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic acids; substituted-5-amino-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acids; substituted-5-amino-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acids; derivatives thereof; pharmaceutical compositions comprising the compounds; and processes for producing the compounds WARNER-LAMBERT COMPANY (US) 1990-02-07 EP disclosed
US-4822801-A 4-oxo-1,4-dihydroquinoline-3-carboxylic acid derivative as antibacterial agents WARNER-LAMBERT COMPANY (US) 1989-04-18 US disclosed
EP-0172651-A1 Substituted-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic acids; substituted-5-amino-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acids; substituted-5-amino-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acids; derivatives thereof; pharmaceutical compositions comprising the compounds; and processes for producing the compounds WARNER-LAMBERT COMPANY (US) 1986-02-26 EP disclosed