SCHEMBL9740877

SCHEMBL9740877

COc1cc2c(cc1OC)CC(=O)N(CC1CCN(CCc3ccc([N+](=O)[O-])cc3)C1)CC2

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 8/20 0.52
ABCG2 Q9UNQ0 7/20 0.52
ACHE P22303 2/20 0.48
BCHE P06276 1/20 0.48
KCNJ1 P48048 3/20 0.45
KCNH2 Q12809 3/20 0.45
MAPT P10636 1/20 0.45
HCN4 Q9Y3Q4 1/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9739245 0.95 ABCG2 (0.51) ABCB1ABCG2ACHEBCHEKCNJ1
Hydrochloric Acid SCHEMBL9740859 0.94 ABCG2 (0.50) ABCB1ABCG2ACHEBCHEKCNJ1
SCHEMBL9739968 0.94 ABCB1 (0.50) ABCB1ABCG2ACHEBCHEKCNJ1
SCHEMBL10720389 0.89 ABCB1 (0.45) ABCB1ABCG2ACHEBCHEKCNJ1
SCHEMBL9739547 0.88 ABCB1 (0.53) ABCB1MAPTHCN4CYP3A4ALOX15
SCHEMBL9739280 0.87 HCN4 (0.59) ABCB1ABCG2KCNH2MAPTHCN4
SCHEMBL9739498 0.83 ABCB1 (0.51) ABCB1MAPTHCN4CYP3A4ALOX15
SCHEMBL9741202 0.83 HCN4 (0.47) ABCB1ABCG2KCNH2MAPTHCN4
SCHEMBL9741588 0.83 HCN4 (0.49) ABCB1ABCG2KCNH2MAPTHCN4
SCHEMBL9739201 0.82 HCN4 (0.49) ABCB1ABCG2ACHEKCNH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0224794-B1 CYCLIC AMINE DERIVATIVES, MEDICINES CONTAINING THESE COMPOUNDS AND PROCESS FOR THEIR PREPARATION Dr. Karl Thomae GmbH (DE) 1990-09-12 EP disclosed
EP-0224794-A2 Cyclic amine derivatives, medicines containing these compounds and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-06-10 EP disclosed