SCHEMBL9744388

SCHEMBL9744388

CCOc1ccc2cc(C#Cc3ccc(-c4ccc(OC)cc4)cc3)ccc2c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.54
CYP11B1 P15538 2/20 0.52
CYP11B2 P19099 2/20 0.52
ESR1 P03372 2/20 0.45
AHR P35869 1/20 0.45
APP P05067 2/20 0.45
CYP19A1 P11511 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
ERN1 O75460 1/20 0.43
NQO1 P15559 1/20 0.42
PDGFRB P09619 1/20 0.42
PDGFRA P16234 1/20 0.42
TUBB4A P04350 1/20 0.42
TUBB P07437 1/20 0.42
TUBA3C P0DPH7 1/20 0.42
TUBA1B P68363 1/20 0.42
TUBA4A P68366 1/20 0.42
TUBB4B P68371 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9741989 0.95 CYP11B1 (0.49) MCHR1CYP11B1CYP11B2ESR1AHR
SCHEMBL9743957 0.94 NQO1 (0.48) MCHR1CYP11B1CYP11B2CYP19A1KDM4E
SCHEMBL9744218 0.91 ESR1 (0.50) MCHR1CYP11B1CYP11B2ESR1AHR
SCHEMBL9742978 0.89 NQO1 (0.54) CYP11B1CYP11B2CYP19A1GAANQO1
SCHEMBL9741991 0.88 MCHR1 (0.58) MCHR1AHRAPPERN1TUBB4A
SCHEMBL9743201 0.88 MCHR1 (0.58) MCHR1CYP11B1CYP11B2AHRAPP
SCHEMBL9743177 0.88 CYP11B1 (0.43) MCHR1CYP11B1CYP11B2CYP19A1KDM4E
SCHEMBL9742321 0.87 APP (0.53) MCHR1CYP11B1CYP11B2APPNQO1
SCHEMBL9743773 0.87 MCHR1 (0.46) MCHR1CYP11B1CYP11B2CYP19A1ALDH1A1
SCHEMBL9743907 0.87 CYP3A4 (0.47) MCHR1CYP11B1CYP11B2CYP19A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084204-A Naphthylacetylenes MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-01-28 US disclosed