SCHEMBL9747909

SCHEMBL9747909

COc1ccc(OCCCCN(C)CCOc2ccc(OC)c(OC)c2)c(C2Sc3ccccc3N(C)C2=O)c1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.51
SMPD1 P17405 2/20 0.41
BCHE P06276 3/20 0.41
RAB9A P51151 1/20 0.40
CACNA1S Q13698 1/20 0.39
ABCB1 P08183 1/20 0.39
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL9748432 0.96 CYP3A4 (0.49) CYP3A4SMPD1BCHERAB9ACACNA1S
Oxalic Acid SCHEMBL7294755 0.90 CYP3A4 (0.49) CYP3A4CACNA1SABCB1
Oxalic Acid SCHEMBL9747733 0.90 CYP3A4 (0.49) CYP3A4CACNA1SABCB1
Hydrochloric Acid SCHEMBL9749787 0.90 CYP3A4 (0.46) CYP3A4SMPD1BCHERAB9ACACNA1S
Hydrochloric Acid SCHEMBL9748803 0.90 CYP3A4 (0.46) CYP3A4SMPD1BCHERAB9ACACNA1S
Oxalic Acid SCHEMBL9748543 0.90 CYP3A4 (0.47) CYP3A4CACNA1SABCB1
SCHEMBL7376974 0.89 CYP3A4 (0.65) CYP3A4BCHECACNA1SACHE
Fumaric Acid SCHEMBL9747504 0.88 CYP3A4 (0.45) CYP3A4ABCB1
Fumaric Acid SCHEMBL9747497 0.88 CYP3A4 (0.45) CYP3A4ABCB1
Hydrochloric Acid SCHEMBL9748141 0.88 CYP3A4 (0.48) CYP3A4SMPD1RAB9ACACNA1SABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0237573-B1 NOVEL BENZOTHIAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1992-01-15 EP claimed
US-4786635-A THERAPEUTIC AGENTS FOR CIRCULATORY DISEASES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1988-11-22 US claimed
EP-0237573-A1 NOVEL BENZOTHIAZINE DERIVATIVES SANTEN PHARMACEUTICAL CO., LTD. (JP) 1987-09-23 EP claimed