SCHEMBL9753355

SCHEMBL9753355

CC(C)c1c(C=CC(O)CC(=O)CC(=O)O)c(-c2ccccc2)nn2cccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.38
MIF P14174 2/20 0.38
KCNH2 Q12809 2/20 0.37
HDAC1 Q13547 2/20 0.37
ADORA2A P29274 3/20 0.36
ADORA1 P30542 3/20 0.36
ADORA2B P29275 2/20 0.36
ADORA3 P0DMS8 2/20 0.36
CYP2C9 P11712 3/20 0.35
KMT2A Q03164 2/20 0.35
PDE4D Q08499 2/20 0.35
MEN1 O00255 1/20 0.35
PDE5A O76074 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
TSHR P16473 1/20 0.35
PDE4A P27815 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753010 0.93 HMGCR (0.40) ADORA3CYP2C9PDE4DALDH1A1CYP3A4
SCHEMBL9753009 0.93 HMGCR (0.40) ADORA3CYP2C9PDE4DALDH1A1CYP3A4
SCHEMBL9753639 0.89 HMGCR (0.34) MIFADORA3CYP2C9PDE4DALDH1A1
SCHEMBL9753646 0.89 HMGCR (0.34) MIFADORA3CYP2C9PDE4DALDH1A1
SCHEMBL9753332 0.86 HMGCR (0.45) ADORA3CYP2C9PDE4DALDH1A1CYP3A4
SCHEMBL9753022 0.84 HMGCR (0.35) ADORA3CYP2C9PDE4DALDH1A1CYP3A4
SCHEMBL9753024 0.84 HMGCR (0.35) ADORA3CYP2C9PDE4DALDH1A1CYP3A4
SCHEMBL9753670 0.83 HMGCR (0.34) ADORA3CYP2C9PDE4DHMGCRABCC3
SCHEMBL9753663 0.83 HMGCR (0.34) ADORA3CYP2C9PDE4DHMGCRABCC3
SCHEMBL9753494 0.81 HMGCR (0.38) ADORA3CYP2C9PDE4DALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed