SCHEMBL9753784

SCHEMBL9753784

Cc1cc(C)n2nc(C(C)C)c(/C=C/C(O)CC(=O)CC(=O)O)c(-c3ccc(F)cc3)c12

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 8/20 0.47
ESR1 P03372 1/20 0.46
CHRM1 P11229 1/20 0.46
TBXA2R P21731 1/20 0.46
PDE4A P27815 1/20 0.46
ADRA1A P35348 1/20 0.46
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
PDE6D O43924 1/20 0.39
NR1I2 O75469 1/20 0.39
PDE4D Q08499 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753794 1.00 HMGCR (0.47) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9753234 0.91 HMGCR (0.47) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9753235 0.91 HMGCR (0.47) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9753373 0.88 HMGCR (0.60) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9753397 0.87 HMGCR (0.48) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9753390 0.87 HMGCR (0.48) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9753589 0.85 HMGCR (0.41) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL9753585 0.85 HMGCR (0.41) HMGCRALDH1A1CYP3A4PDE6DNR1I2
SCHEMBL9753337 0.80 HMGCR (0.48) HMGCRESR1CHRM1TBXA2RPDE4A
SCHEMBL9753329 0.80 HMGCR (0.48) HMGCRESR1CHRM1TBXA2RPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018903-A1 PYRROLOPYRIDAZINE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-12 WO disclosed