SCHEMBL9753984

SCHEMBL9753984

CCCCC(=O)C(Cc1ccc(-c2ccccc2C#N)cc1)/C(=N/OC)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MME P08473 1/20 0.44
FFAR1 O14842 1/20 0.44
AKR1B1 P15121 1/20 0.44
PTPN1 P18031 1/20 0.40
ITGB1 P05556 1/20 0.40
ITGA4 P13612 1/20 0.40
TSHR P16473 1/20 0.39
GRIA2 P42262 1/20 0.39
GRIA4 P48058 1/20 0.39
LTB4R2 Q9NPC1 7/20 0.37
AGTR1 P30556 1/20 0.37
AGTR2 P50052 1/20 0.37
ACHE P22303 1/20 0.36
ESR2 Q92731 1/20 0.35
PPARG P37231 2/20 0.35
PPARA Q07869 1/20 0.35
EGLN1 Q9GZT9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9753986 1.00 MME (0.44) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL7815803 0.90 MME (0.40) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL7815799 0.90 MME (0.40) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL2572010 0.86 MME (0.52) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL633444 0.84 MME (0.48) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL9710320 0.83 MME (0.51) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL1895025 0.82 MME (0.46) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL9710577 0.82 MME (0.50) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL9710219 0.82 MME (0.50) MMEFFAR1AKR1B1PTPN1ITGB1
SCHEMBL1371403 0.81 MME (0.48) MMEFFAR1AKR1B1PTPN1ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991015479-A1 SUBSTITUTED PYRAZOLES, ISOXAZOLES AND ISOTHIAZOLES MERCK & CO., INC. (US) 1991-10-17 WO disclosed