Tryptoline

Tryptoline

SCHEMBL9754749

c1ccc2c3c([nH]c2c1)CNCC3.c1ccc2c3c([nH]c2c1)CNCC3.c1ccc2c3c([nH]c2c1)CNCC3

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 3/20 1.00
KDM4E B2RXH2 3/20 1.00
NR2E1 Q9Y466 2/20 1.00
HTR5A P47898 1/20 1.00
HTR2A P28223 1/20 0.77
HTR2C P28335 1/20 0.77
TAAR1 Q96RJ0 1/20 0.72
CYP1A2 P05177 2/20 0.56
ADRA2A P08913 1/20 0.56
ADRA2B P18089 1/20 0.56
ADRA2C P18825 1/20 0.56
HTR7 P34969 1/20 0.56
LMNA P02545 1/20 0.56
CYP2D6 P10635 1/20 0.56
THRB P10828 1/20 0.56
ALOX15 P16050 1/20 0.56
TSHR P16473 1/20 0.56
NFKB1 P19838 1/20 0.56
RECQL P46063 1/20 0.56
PMP22 Q01453 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tryptoline SCHEMBL171755 1.00 NISCH (1.00) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL9480983 1.00 NISCH (1.00) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL12190178 1.00 NISCH (1.00) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL29350043 1.00 NISCH (1.00) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL30213301 0.98 NISCH (0.96) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL8818317 0.98 NISCH (0.96) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL28226558 0.98 NISCH (0.96) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL28477910 0.96 NISCH (0.93) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL29139386 0.92 NISCH (0.84) NISCHKDM4ENR2E1HTR5AHTR2A
Tryptoline SCHEMBL28856564 0.91 NISCH (0.82) NISCHKDM4ENR2E1HTR5AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991014184-A1 BETA CARBOLINES AS VITAL STAINS FOR NEUROTRANSMITTER SYSTEMS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1991-09-19 WO disclosed