SCHEMBL9756772

SCHEMBL9756772

CC(C)c1c(/C=C/C(O)CC(=O)CC(=O)O)c(-c2ccc(F)cc2)c(-c2ccccc2)n1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 10/20 0.48
ABCB11 O95342 3/20 0.45
SLCO1B1 Q9Y6L6 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
NR1I2 O75469 1/20 0.45
RHOC P08134 1/20 0.45
CYP3A4 P08684 1/20 0.45
THRB P10828 1/20 0.45
NR1H4 Q96RI1 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.45
CYP2C9 P11712 3/20 0.42
SIRT6 Q8N6T7 2/20 0.42
ABCC3 O15438 2/20 0.42
PGR P06401 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
RXRA P19793 1/20 0.42
TBXA2R P21731 1/20 0.42
CCKAR P32238 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10650833 0.92 HMGCR (0.46) HMGCRABCB11SLCO1B1HDAC1HDAC2
SCHEMBL9773648 0.86 HMGCR (0.42) HMGCRABCB11SLCO1B1HDAC1HDAC2
SCHEMBL9773646 0.86 HMGCR (0.42) HMGCRABCB11SLCO1B1HDAC1HDAC2
SCHEMBL9773769 0.85 HMGCR (0.41) HMGCRABCB11SLCO1B1HDAC1HDAC2
SCHEMBL9756757 0.84 HMGCR (0.56) HMGCRTBXA2RADRA1A
SCHEMBL9665214 0.81 HMGCR (0.42) HMGCRABCB11CYP2C9SIRT6ABCC3
SCHEMBL9665217 0.81 HMGCR (0.42) HMGCRABCB11CYP2C9SIRT6ABCC3
SCHEMBL9662629 0.81 HMGCR (0.53) HMGCRABCB11CYP2C9SIRT6ABCC3
SCHEMBL9662639 0.81 HMGCR (0.53) HMGCRABCB11CYP2C9SIRT6ABCC3
SCHEMBL9773771 0.81 HMGCR (0.40) HMGCRABCB11SLCO1B1HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4992462-A Inhibitor of HMG-CoA reductase BAYER AKTIENGESELLSCHAFT (DE) 1991-02-12 US disclosed