Bromide

Bromide

SCHEMBL9757461

Br.CSC(C)Cn1c(=N)sc2cc(OC(F)(F)F)ccc21

nearest known ligand 0.40

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 1/20 0.34
SLC6A3 known ✓ Q01959 1/20 0.34
KCNQ3 O43525 16/20 0.40
KCNQ2 O43526 16/20 0.40
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
GMNN O75496 1/20 0.34
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
GAA P10253 1/20 0.34
CYP2C9 P11712 1/20 0.34
PKM P14618 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650311 0.99 KCNQ3 (0.40) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
SCHEMBL9780567 0.83 KCNQ3 (0.40) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
SCHEMBL8651427 0.82 KCNQ3 (0.43) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL9757631 0.81 KCNQ3 (0.42) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
SCHEMBL8661581 0.81 KCNQ3 (0.39) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
SCHEMBL9757555 0.81 KCNQ3 (0.41) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
SCHEMBL1393108 0.80 SMN1; SMN2 (0.43) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL9780209 0.79 SMN1; SMN2 (0.43) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
SCHEMBL9471831 0.79 SMN1; SMN2 (0.42) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL6255293 0.79 SMN1; SMN2 (0.42) KCNQ3KCNQ2SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008280-A Treatment of glutamate-induced convulsions, schizophrenia RHONE-POULENC SANTE (FR) 1991-04-16 US disclosed