SCHEMBL9763463

SCHEMBL9763463

CN(CCN(C)C(=O)c1cccnc1)C(=O)c1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.56
ALDH1A1 P00352 3/20 0.53
GAA P10253 2/20 0.53
APP P05067 1/20 0.53
HCAR3 P49019 1/20 0.53
HCAR2 Q8TDS4 1/20 0.53
HSD17B10 Q99714 3/20 0.52
TSHR P16473 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
ALOX15 P16050 2/20 0.52
USP2 O75604 1/20 0.52
TP53 P04637 1/20 0.52
MAPK1 P28482 1/20 0.52
F7 P08709 1/20 0.52
F3 P13726 1/20 0.52
SARM1 Q6SZW1 1/20 0.52
SIRT2 Q8IXJ6 1/20 0.52
SIRT6 Q8N6T7 1/20 0.52
SIRT1 Q96EB6 1/20 0.52
SIRT3 Q9NTG7 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15477469 0.95 HTT (0.52) HTTALDH1A1GAAAPPHCAR3
SCHEMBL31707265 0.92 HTT (0.52) HTTALDH1A1GAAAPPHCAR3
SCHEMBL24508715 0.92 HTT (0.52) HTTALDH1A1GAAAPPHCAR3
SCHEMBL16435722 0.89 KDM4E (0.49) HTTALDH1A1GAAAPPHCAR3
SCHEMBL30476608 0.88 HTT (0.63) HTTALDH1A1GAAAPPHCAR3
SCHEMBL27670331 0.88 HTT (0.55) HTTALDH1A1GAAAPPHCAR3
SCHEMBL2111661 0.88 HTT (0.63) HTTALDH1A1GAAAPPHCAR3
SCHEMBL31277621 0.88 HTT (0.49) HTTALDH1A1GAAAPPHCAR3
Hydrochloric Acid SCHEMBL30055763 0.86 HTT (0.61) HTTALDH1A1GAAAPPHCAR3
SCHEMBL24970247 0.85 HTT (0.52) HTTALDH1A1GAAAPPHCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4994462-A N,N-Bis(nipecotyl)piperazines RESEARCH CORPORATION (US) 1991-02-19 US disclosed
US-4798830-A TETRAHYDROQUINOLINE DERIVATIVES RESEARCH CORPORATION (US) 1989-01-17 US disclosed
US-4634709-A PIPERIDINE DERIVATIVES RESEARCH CORPORATION (US) 1987-01-06 US disclosed
US-4443450-A N,N*-BIS(NIPECOTYL) PIPERAZINE RESEARCH CORPORATION (US) 1984-04-17 US disclosed