SCHEMBL9765669

SCHEMBL9765669

CCCn1c(=O)n(C)c(=O)c2[nH]cnc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 18/20 1.00
PDE4B Q07343 18/20 1.00
PDE4C Q08493 18/20 1.00
PDE4D Q08499 18/20 1.00
ADORA2A P29274 12/20 1.00
ADORA2B P29275 8/20 1.00
PDE2A O00408 1/20 0.69
PDE5A O76074 1/20 0.69
CYP1A2 P05177 1/20 0.69
CYP3A4 P08684 1/20 0.69
CFTR P13569 1/20 0.69
TSHR P16473 1/20 0.69
MAPK1 P28482 1/20 0.69
ADORA1 P30542 1/20 0.69
SCN1A P35498 1/20 0.69
PDE6C P51160 1/20 0.69
PDE1A P54750 1/20 0.69
PDE1B Q01064 1/20 0.69
PDE3B Q13370 1/20 0.69
PDE7A Q13946 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1331789 0.91 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL515771 0.90 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3177911 0.90 PDE4A (0.92) PDE4APDE4BPDE4CPDE4DADORA2A
Ammonia Solution, Strong SCHEMBL10420651 0.89 PDE4A (0.97) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381254 0.88 PDE4A (0.89) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL4623455 0.88 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
Water SCHEMBL27461178 0.88 ADORA2A (0.97) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7460178 0.88 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL5400933 0.86 PDE4A (0.91) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL21381259 0.85 PDE4A (1.00) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3220190-A None JP disclosed
JP-H03220190-A XANTHINE COMPOUND HOKURIKU SEIYAKU CO LTD 1991-09-27 JP disclosed