SCHEMBL9765788

SCHEMBL9765788

CC1=C(C(=O)OCC2COC(C)(C)O2)C(c2cccc([N+](=O)[O-])c2)C(C(=O)OC(C)C)=C(C)N1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.68
CYP1A2 P05177 4/20 0.68
CYP3A4 P08684 4/20 0.68
CYP2C9 P11712 4/20 0.68
CYP2C19 P33261 4/20 0.68
KMT2A Q03164 4/20 0.68
LMNA P02545 3/20 0.68
MAPT P10636 3/20 0.68
CYP2D6 P10635 2/20 0.68
TSHR P16473 2/20 0.68
NFKB1 P19838 2/20 0.68
THPO P40225 2/20 0.68
CACNA1F O60840 9/20 0.64
CACNA1D Q01668 9/20 0.64
CACNA1S Q13698 9/20 0.64
CACNA1C Q13936 9/20 0.64
ADORA3 P0DMS8 2/20 0.61
NR1I2 O75469 1/20 0.58
NR3C1 P04150 1/20 0.58
ABCB1 P08183 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10391379 0.95 CACNA1F (0.68) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9765779 0.92 CACNA1F (0.73) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10391383 0.91 CACNA1F (0.63) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9765716 0.91 HIF1A (0.70) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10391380 0.91 CACNA1F (0.63) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10503328 0.84 CACNA1C (0.65) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL9505209 0.84 CACNA1F (0.87) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL11011759 0.83 MEN1 (0.82) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10721143 0.83 CACNA1F (0.59) MEN1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL10391543 0.83 HIF1A (0.66) MEN1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4988717-A Optically active 1,4-dihydropyridine esters useful for treating circulatory illnesses BAYER AKTIENGESELLSCHAFT (DE) 1991-01-29 US disclosed
US-4849433-A The compound, (⃡)1,4-dihydro-2,6-dimethyl-4-(2'-nitrophenyl)-pyridine-3,5-dicarboxylic acid, methyl isobutyl ester, compositions containing same and a method for effecting coronary dilation BAYER AKTIENGESELLSCHAFT (DE) 1989-07-18 US disclosed
US-4510310-A 1,4-Dihydro-2,6-dimethyl-4-(2'-chlorophenyl)-3,5-dicarboxylic acid,methyl or ethyl,trifluoroethyl ester BAYER AKTIENGESELLSCHAFT (DE) 1985-04-09 US disclosed