SCHEMBL9776705

SCHEMBL9776705

Cc1ccccc1Nc1nc(N(C)c2ccccc2)c2ccccc2n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.59
LMNA P02545 1/20 0.59
PKM P14618 1/20 0.59
NFKB1 P19838 1/20 0.59
RAB9A P51151 1/20 0.59
NFKB2 Q00653 1/20 0.59
RELA Q04206 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9776921 0.99 NPC1 (0.61) NPC1LMNAPKMNFKB1RAB9A
Hydrochloric Acid SCHEMBL9776836 0.99 NPC1 (0.61) NPC1LMNAPKMNFKB1RAB9A
Hydrochloric Acid SCHEMBL9776694 0.90 NPC1 (0.55) NPC1LMNAPKMNFKB1RAB9A
Hydrochloric Acid SCHEMBL9776710 0.88 EGFR (0.63)
Hydrochloric Acid SCHEMBL9776722 0.86 NPC1 (0.66) NPC1LMNAPKMNFKB1RAB9A
SCHEMBL9776764 0.85
SCHEMBL9508870 0.85
Hydrochloric Acid SCHEMBL9776934 0.84
Hydrochloric Acid SCHEMBL9776718 0.84
Hydrochloric Acid SCHEMBL9811774 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5064833-A Substituted quinazoline derivatives for use in gastrointestinal diseases SMITHKLINE BEECHAM INTERCREDIT B.V. (GB) 1991-11-12 US claimed
EP-0322133-B1 QUINAZOLINE DERIVATIVES SmithKline Beecham Intercredit B.V. (NL) 1991-05-22 EP claimed
EP-0322133-A1 Quinazoline derivatives SmithKline Beecham Intercredit B.V. (NL) 1989-06-28 EP claimed