SCHEMBL978266

SCHEMBL978266

COc1ccc(-c2ccc3cc(C(=O)O)ccc3c2)cc1OC

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 5/20 0.72
RARG P13631 5/20 0.72
RARA P10276 4/20 0.72
CA12 O43570 1/20 0.69
CA1 P00915 1/20 0.69
CA2 P00918 1/20 0.69
CA4 P22748 1/20 0.69
CA6 P23280 1/20 0.69
CA7 P43166 1/20 0.69
TPMT P51580 1/20 0.69
CA9 Q16790 1/20 0.69
CA14 Q9ULX7 1/20 0.69
LMNA P02545 3/20 0.61
MEN1 O00255 1/20 0.61
NR1I2 O75469 1/20 0.61
PGR P06401 1/20 0.61
HSPD1 P10809 1/20 0.61
GOT1 P17174 1/20 0.61
GLRA1 P23415 1/20 0.61
BLM P54132 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2040708 0.86 CA12 (0.72) RARBRARGRARACA12CA1
SCHEMBL4946900 0.84 KDM4E (0.70) RARBRARGRARACA12CA1
SCHEMBL980501 0.84 RARB (1.00) RARBRARGRARACA12CA1
SCHEMBL30301169 0.84 RARB (1.00) RARBRARGRARACA12CA1
SCHEMBL5047379 0.83 KDM4E (0.74) RARBRARGRARACA1CA2
Veratric Acid SCHEMBL29386353 0.82 CA12 (1.00) CA12CA1CA2CA4CA6
Veratric Acid SCHEMBL114848 0.82 CA12 (1.00) CA12CA1CA2CA4CA6
Veratric Acid SCHEMBL976032 0.82 CA12 (1.00) CA12CA1CA2CA4CA6
SCHEMBL13900230 0.82 RARB (0.64) RARBRARGRARALMNAMEN1
SCHEMBL6244003 0.82 CA12 (0.71) RARBRARGRARACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150098918-A1 CREAM GELS COMPRISING AT LEAST ONE RETINOID AND BENZOYL PEROXIDE GALDERMA RESEARCH & DEVELOPMENT (FR) 2015-04-09 US claimed
US-20100166852-A1 Cream gels comprising at least one retinoid and benzoyl peroxide GALDERMA RESEARCH & DEVELOPMENT (FR) 2010-07-01 US claimed
US-20090318550-A1 Emulsions comprising at least one retinoid and benzoyl peroxide GALDERMA RESEARCH & DEVELOPMENT (FR) 2009-12-24 US claimed
US-RE34805-E Treatment of dermatologic diseases, degeneration of conjunctive tissues; antitumor activity CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (CIRD) (FR) 1994-12-06 US claimed
US-4940696-A Benzonaphthalene derivatives and their use in therapeutic and cosmetic compositions CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIOUES (CIRD) (FR) 1990-07-10 US claimed
EP-0199636-B1 BENZONAPHTHALENIC DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN PHARMACY AND COSMETICS CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES C.I.R.D. Groupement d'Intérêt Economique dit: (FR) 1989-02-08 EP claimed
US-10925814-B2 Cream gels comprising at least one retinoid and benzoyl peroxide GALDERMA RESEARCH & DEVELOPMENT (FR) 2021-02-23 US disclosed
US-10702466-B2 Emulsions comprising at least one retinoid and benzoyl peroxide GALDERMA RESEARCH & DEVELOPMENT (FR) 2020-07-07 US disclosed
US-20180263865-A1 CREAM GELS COMPRISING AT LEAST ONE RETINOID AND BENZOYL PEROXIDE GALDERMA RESEARCH & DEVELOPMENT (FR) 2018-09-20 US disclosed
US-9999577-B2 Cream gels comprising at least one retinoid and benzoyl peroxide GALDERMA RESEARCH & DEVELOPMENT (FR) 2018-06-19 US disclosed
EP-3184108-A1 COMPOSITION COMPRISING A RETINOID AND BENZOYL PEROXIDE Galderma Research & Development (FR) 2017-06-28 EP disclosed
US-9060948-B2 Dermatological/cosmetic compositions comprising a retinoid and benzoyl peroxide GALDERMA RESEARCH & DEVELOPMENT (FR) 2015-06-23 US disclosed
US-20150098918-A1 CREAM GELS COMPRISING AT LEAST ONE RETINOID AND BENZOYL PEROXIDE GALDERMA RESEARCH & DEVELOPMENT (FR) 2015-04-09 US disclosed
US-RE34805-E Treatment of dermatologic diseases, degeneration of conjunctive tissues; antitumor activity CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (CIRD) (FR) 1994-12-06 US disclosed
US-RE34440-E Treatment of dermatological diseases and degeneration of conjunctive tissues; antitumor agent CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1993-11-09 US disclosed
US-5212303-A Benzonaphthalene derivatives, a process for their preparation and their use in therapeutic and cosmetic compositions CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (CIRD) (FR) 1993-05-18 US disclosed
US-5183889-A For topical or systemic treatment of dermatologic disease, degeneration of conjunction tissues and tumors CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (CIRD) (FR) 1993-02-02 US disclosed
US-5098895-A Skin disorders and antitumor agents CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1992-03-24 US disclosed
US-4940696-A Benzonaphthalene derivatives and their use in therapeutic and cosmetic compositions CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIOUES (CIRD) (FR) 1990-07-10 US disclosed
US-4717720-A DERMATOLOGIC DISEASES, CONJUCTIVE TISSUE DEGENERATION AND ANTI-TUMOR ACTIVITY CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES (C.I.R.D.) (FR) 1988-01-05 US disclosed