SCHEMBL9788773

SCHEMBL9788773

CCc1ccc(-c2ccc(-c3nc4ccccc4c(C(=O)O)c3C)cc2)cc1

nearest known ligand 0.80

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 15/20 0.80
PDE10A Q9Y233 3/20 0.79
TSHR P16473 1/20 0.74
KMT2A Q03164 1/20 0.56
LMNA P02545 1/20 0.56
POLB P06746 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1581468 0.86 PDE10A (1.00) DHODHPDE10ATSHRKMT2ALMNA
Hydrochloric Acid SCHEMBL27511204 0.84 PDE10A (0.97) DHODHPDE10ATSHRKMT2ALMNA
SCHEMBL17593892 0.84 DHODH (0.68) DHODHPDE10ATSHR
SCHEMBL13529075 0.81 DHODH (0.76) DHODHPDE10A
SCHEMBL5205114 0.78 PDE10A (0.68) DHODHPDE10ATSHR
SCHEMBL14492079 0.77 PDE10A (0.68) DHODHPDE10ATSHRLMNAPOLB
SCHEMBL9052974 0.77 DHODH (0.68) DHODHPDE10ATSHR
SCHEMBL3234894 0.76 KDM4E (0.68) DHODHPDE10ATSHRKMT2ALMNA
SCHEMBL2372674 0.75 PDE10A (0.73) DHODHPDE10ATSHRKMT2ALMNA
SCHEMBL4879923 0.75 PDE10A (0.72) DHODHPDE10ATSHRKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032597-A Antitumor DU PONT MERCK PHARMACEUTICAL (US) 1991-07-16 US disclosed
EP-0133244-B1 PHENYLQUINOLINECARBOXYLIC ACIDS AND DERIVATIVES AS ANTITUMOR AGENTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1990-12-05 EP disclosed
US-4680299-A ANTITUMOR AGENTS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1987-07-14 US disclosed
EP-0133244-A2 Phenylquinolinecarboxylic acids and derivatives as antitumor agents E.I. DU PONT DE NEMOURS AND COMPANY (US) 1985-02-20 EP disclosed