SCHEMBL9795396

SCHEMBL9795396

CC(C(=O)c1ccccc1)n1cncn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.49
KMT2A Q03164 4/20 0.48
HSP90AA1 P07900 2/20 0.48
MAPT P10636 1/20 0.48
LMNA P02545 2/20 0.47
TSHR P16473 1/20 0.46
CYP26A1 O43174 3/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ALDH1A1 P00352 3/20 0.43
GAA P10253 1/20 0.43
PGR P06401 1/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
HTR2A P28223 1/20 0.42
HRH1 P35367 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9199550 0.86 KMT2A (0.64) CYP19A1KMT2AHSP90AA1MAPTLMNA
SCHEMBL6227295 0.84 CYP19A1 (0.51) CYP19A1KMT2AHSP90AA1MAPTLMNA
SCHEMBL10361474 0.84 HSP90AA1 (0.49) CYP19A1KMT2AHSP90AA1MAPTCYP26A1
Hydrochloric Acid SCHEMBL9792757 0.83 HSP90AA1 (0.48) CYP19A1KMT2AHSP90AA1MAPTCYP26A1
SCHEMBL11563115 0.81 CYP19A1 (0.50) CYP19A1KMT2AHSP90AA1MAPTLMNA
SCHEMBL10361626 0.81 HSP90AA1 (0.49) CYP19A1KMT2AHSP90AA1MAPTCYP26A1
SCHEMBL10711903 0.81 CYP19A1 (0.53) CYP19A1KMT2AHSP90AA1MAPTLMNA
SCHEMBL10408460 0.79 CYP19A1 (0.56) CYP19A1KMT2AHSP90AA1MAPTLMNA
SCHEMBL10568532 0.79 HSP90AA1 (0.47) KMT2AHSP90AA1LMNACYP26A1CYP3A4
SCHEMBL10570329 0.78 SLC6A4 (0.43) CYP19A1KMT2AHSP90AA1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5032607-A Enzyme inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-07-16 US disclosed
US-4945101-A Fungicidal novel hydroxyalkynyl-azolyl derivatives BAYER AKTIENGESELLSCHAFT (DE) 1990-07-31 US disclosed
US-4866086-A PHENYLTRIAZOLYL OLEFINIC AROMATASE INHIBITORS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-09-12 US disclosed
EP-0192055-B1 HYDROXYALKYNYL-AZOLYL DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS FUNGICIDES BAYER AG (DE) 1989-08-09 EP disclosed
EP-0299683-A2 Heterocyclic olefinic compounds and their use as aromatase inhibitors IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-01-18 EP disclosed
US-4625036-A Antifungal azole compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1986-11-25 US disclosed
EP-0192055-A2 Hydroxyalkynyl-azolyl derivatives, process for their preparation and their use as fungicides BAYER AG (DE) 1986-08-27 EP disclosed
US-4578396-A Fungicidal hydroxyalkinyl-azolyl derivatives BAYER AKTIENGESELLSCHAFT (DE) 1986-03-25 US disclosed
EP-0122693-A1 Antifungal di(azolyl)propanol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-10-24 EP disclosed
EP-0096786-A2 Hydroxyalkynyl-azolyl derivatives, process for their preparation and their use as fungicides BAYER AG (DE) 1983-12-28 EP disclosed