SCHEMBL9799082

SCHEMBL9799082

Cc1cc(Cn2cnc3c(Cl)nc(N)nc32)c(C)s1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 20/20 0.59
HSP90AA1 P07900 19/20 0.59
HSP90B1 P14625 1/20 0.52
TRAP1 Q12931 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9798287 0.80 PNP (0.57) HSP90AB1HSP90AA1
SCHEMBL3396283 0.79 HSP90AB1 (0.64) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL14568306 0.78 HSP90AB1 (0.77) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3396202 0.77 HSP90AB1 (0.73) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3392317 0.76 HSP90AB1 (0.58) HSP90AB1HSP90AA1
SCHEMBL3393055 0.76 HSP90AB1 (0.54) HSP90AB1HSP90AA1
SCHEMBL3396492 0.76 HSP90AB1 (0.76) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL27854926 0.75 CDK1 (0.71) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3396346 0.75 HSP90AB1 (0.67) HSP90AB1HSP90AA1
SCHEMBL3396801 0.75 HSP90AB1 (0.71) HSP90AB1HSP90AA1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5051429-A For treatment of autoimmune diseases such as arthritis, lupus, antiinflammatory agents, multiple sclerosis, diabetes and viral diseases WARNER-LAMBERT CO. (US) 1991-09-24 US disclosed
US-4952693-A TREATING AUTOIMMUNE DISEASES WARNER-LAMBERT COMPANY (US) 1990-08-28 US disclosed
US-4772606-A AUTOIMMUNE DISEASES, ORGAN TRANSPLANTS WARNER-LAMBERT COMPANY (US) 1988-09-20 US disclosed
EP-0178178-A2 Purine derivatives WARNER-LAMBERT COMPANY (US) 1986-04-16 EP disclosed