SCHEMBL9803307

SCHEMBL9803307

CCN1CCCC1CCNCC(=O)N1c2ccccc2C(=O)Nc2cccnc21

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.63
CYP1A2 P05177 1/20 0.63
CYP3A4 P08684 1/20 0.63
CHRM4 P08173 1/20 0.63
CHRM1 P11229 1/20 0.63
CHRM3 P20309 1/20 0.63
MAPK1 P28482 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9803358 0.99 CHRM2 (0.62) CHRM2CYP1A2CYP3A4CHRM4CHRM1
SCHEMBL9803038 0.91 CHRM2 (0.62) CHRM2CYP1A2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL10529214 0.90 CHRM2 (0.61) CHRM2CHRM4CHRM1
SCHEMBL10512469 0.89 CHRM2 (0.62) CHRM2CYP1A2CYP3A4CHRM4CHRM1
SCHEMBL9871420 0.86 CHRM2 (0.65) CHRM2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL9879815 0.85 CHRM2 (0.64) CHRM2CHRM4CHRM1CHRM3
SCHEMBL8881347 0.84 CHRM2 (0.66) CHRM2CYP1A2CYP3A4CHRM4CHRM1
SCHEMBL11445770 0.84 CHRM2 (0.63) CHRM2CYP1A2CHRM4CHRM1CHRM3
Hydrochloric Acid SCHEMBL10513989 0.84 CHRM2 (0.61) CHRM2CHRM4CHRM1
SCHEMBL9803290 0.84 CYP1A2 (0.69) CHRM2CYP1A2CYP3A4CHRM4CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026699-A Antiarrhythmia agents DR. KARL THOMAE GMBH (DE) 1991-06-25 US disclosed
US-5002943-A Antispasmodic Agents, Bradycardia Treatment MIHM GERHARD (DE) 1991-03-26 US disclosed
EP-0346745-A1 Condensed diazepinones, processes for their preparation and pharmaceutical preparations containing them Dr. Karl Thomae GmbH (DE) 1989-12-20 EP disclosed