SCHEMBL9817864

SCHEMBL9817864

C#Cc1cccc(Oc2ccc(S(=O)(=O)c3ccc(Oc4cccc(C#C)c4)cc3)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
TDP1 Q9NUW8 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.50
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA9 Q16790 2/20 0.47
CA14 Q9ULX7 1/20 0.47
HAO1 Q9UJM8 1/20 0.43
SOS1 Q07889 1/20 0.42
PGR P06401 2/20 0.41
EGFR P00533 1/20 0.41
FFAR1 O14842 1/20 0.39
POLB P06746 1/20 0.39
APEX1 P27695 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
LMNA P02545 1/20 0.39
ALDH1A1 P00352 2/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11292405 1.00 HTT (0.56) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11301335 1.00 HTT (0.56) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11294599 0.98 HTT (0.55) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11300230 0.98 HTT (0.55) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11300232 0.98 HTT (0.55) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11298933 0.97 HTT (0.54) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11298696 0.97 HTT (0.54) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11301110 0.97 HTT (0.54) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11298929 0.95 HTT (0.52) HTTL3MBTL1TDP1SMN1; SMN2CA12
SCHEMBL11519808 0.95 HTT (0.54) HTTL3MBTL1TDP1SMN1; SMN2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0169205-B1 METHOD OF PREPARING COPOLYMERS UTILIZING ISOIMIDES Hughes Aircraft Company (US) 1991-11-13 EP claimed
US-4613637-A COATINGS, FILMS, ENCAPSULANTS HUGHES AIRCRAFT COMPANY (US) 1986-09-23 US claimed
EP-0169205-A1 METHOD OF PREPARING COPOLYMERS UTILIZING ISOIMIDES. HUGHES AIRCRAFT CO (US) 1986-01-29 EP claimed
WO-1985002853-A1 COPOLYMERS UTILIZING ISOIMIDES AND METHOD OF PREPARING SAME HUGHES AIRCRAFT COMPANY (US) 1985-07-04 WO claimed
US-4131625-A REACTIVE PLASTICIZER FOR POLYSULFONES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1978-12-26 US claimed
US-4108926-A 4,4*-BIS(3-ETHYNYLPHENOXY)DIPHENYL SULFONE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1978-08-22 US claimed
EP-0169205-B1 METHOD OF PREPARING COPOLYMERS UTILIZING ISOIMIDES Hughes Aircraft Company (US) 1991-11-13 EP disclosed
US-4837256-A SOLVENT RESISTANCE AMOCO CORPORATION (US) 1989-06-06 US disclosed
US-4613637-A COATINGS, FILMS, ENCAPSULANTS HUGHES AIRCRAFT COMPANY (US) 1986-09-23 US disclosed
US-4587315-A Diethynylated phenylbenzimidazole compounds HUGHES AIRCRAFT COMPANY (US) 1986-05-06 US disclosed
EP-0169205-A1 METHOD OF PREPARING COPOLYMERS UTILIZING ISOIMIDES. HUGHES AIRCRAFT CO (US) 1986-01-29 EP disclosed
US-4537974-A Diethynylated phenylbenzimidazole compounds HUGHES AIRCRAFT COMPANY (US) 1985-08-27 US disclosed
WO-1985002853-A1 COPOLYMERS UTILIZING ISOIMIDES AND METHOD OF PREPARING SAME HUGHES AIRCRAFT COMPANY (US) 1985-07-04 WO disclosed
US-4417039-A Cis-enyne aromatic and aromatic heterocyclic polymers THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1983-11-22 US disclosed
US-4356325-A Process for preparation of acetylene terminated sulfones, oligomers and precursors therefor GULF RESEARCH & DEVELOPMENT COMPANY (US) 1982-10-26 US disclosed
US-4131625-A REACTIVE PLASTICIZER FOR POLYSULFONES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1978-12-26 US disclosed
US-4131625-A REACTIVE PLASTICIZER FOR POLYSULFONES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1978-12-26 US disclosed
US-4131625-A REACTIVE PLASTICIZER FOR POLYSULFONES THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1978-12-26 US disclosed
US-4108926-A 4,4*-BIS(3-ETHYNYLPHENOXY)DIPHENYL SULFONE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1978-08-22 US disclosed
US-4108926-A 4,4*-BIS(3-ETHYNYLPHENOXY)DIPHENYL SULFONE THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE AIR FORCE (US) 1978-08-22 US disclosed