SCHEMBL9825129

SCHEMBL9825129

NC(=O)[C@H]1CN(CCC2COc3ccccc3O2)CC[C@H]1N

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.48
ALOX5 P09917 1/20 0.46
HTR1A P08908 2/20 0.44
ADRA2A P08913 1/20 0.43
DRD1 P21728 1/20 0.43
TBXA2R P21731 1/20 0.43
SLC6A2 P23975 1/20 0.43
ADRA1A P35348 1/20 0.43
DRD3 P35462 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9826185 1.00 HTT (0.48) HTTALOX5HTR1AADRA2ADRD1
SCHEMBL9825132 1.00 HTT (0.48) HTTALOX5HTR1AADRA2ADRD1
SCHEMBL9826195 1.00 HTT (0.48) HTTALOX5HTR1AADRA2ADRD1
SCHEMBL9692523 1.00 HTT (0.48) HTTALOX5HTR1AADRA2ADRD1
SCHEMBL9824754 0.84 HTT (0.46) HTTALOX5HTR1A
SCHEMBL9825951 0.84 HTT (0.46) HTTALOX5HTR1A
SCHEMBL9825683 0.82 HTT (0.48) HTTHTR1A
SCHEMBL9692391 0.78 HTT (0.48) HTTHTR1AADRA1A
SCHEMBL9692374 0.78 HTT (0.48) HTTHTR1AADRA1A
SCHEMBL9692630 0.78 HTT (0.46) HTTHTR1AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP claimed