SCHEMBL9832017

SCHEMBL9832017

CCOC(=O)C1(CC)C(=O)Nc2cc(NC(=O)c3cccnc3)c([N+](=O)[O-])cc21

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.51
NPC1 O15118 1/20 0.51
TP53 P04637 1/20 0.45
ALDH1A1 P00352 6/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
KMT2A Q03164 1/20 0.41
ABCB1 P08183 1/20 0.41
ABCC1 P33527 1/20 0.41
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CYP2C19 P33261 1/20 0.40
GFER P55789 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831754 0.97 MAPT (0.51) MAPTNPC1TP53ALDH1A1KDM4E
SCHEMBL9832723 0.90 MAPT (0.40) MAPTNPC1ALDH1A1KDM4EMEN1
SCHEMBL9831567 0.89 MAPT (0.52) MAPTNPC1TP53ALDH1A1KDM4E
SCHEMBL9831783 0.86 MAPT (0.39) MAPTNPC1ALDH1A1KDM4EMEN1
SCHEMBL9833516 0.86 MAPT (0.52) MAPTNPC1TP53ALDH1A1KDM4E
SCHEMBL11025025 0.85 MAPT (0.38) MAPTNPC1TP53ALDH1A1KDM4E
SCHEMBL11023012 0.82 MAPT (0.38) MAPTNPC1TP53ALDH1A1KDM4E
SCHEMBL9832729 0.82 MAPT (0.57) MAPTNPC1ALDH1A1KDM4EMEN1
SCHEMBL9833125 0.82 MAPT (0.54) MAPTNPC1TP53ALDH1A1MEN1
SCHEMBL9831749 0.80 MAPT (0.54) MAPTNPC1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed