SCHEMBL9832844

SCHEMBL9832844

COC(=O)C1(C)C(=O)Nc2cc3c(cc21)NC(c1cccnc1)N3

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.40
MAPT P10636 3/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
RAB9A P51151 2/20 0.40
MAPK1 P28482 1/20 0.40
RECQL P46063 1/20 0.40
MCL1 Q07820 1/20 0.40
TSHR P16473 3/20 0.39
HTT P42858 1/20 0.38
GAA P10253 5/20 0.37
CYP2C9 P11712 4/20 0.37
CYP1A2 P05177 2/20 0.37
ALDH1A1 P00352 5/20 0.37
HPGD P15428 3/20 0.37
HSD17B10 Q99714 2/20 0.37
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
CYP3A4 P08684 4/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833624 0.89 KDM4E (0.46) KDM4EMAPTMEN1KMT2ARAB9A
SCHEMBL9834043 0.88 KDM4E (0.42) KDM4EMAPTMEN1KMT2ARAB9A
SCHEMBL9832551 0.88 KDM4E (0.39) KDM4EMAPTMEN1KMT2AMAPK1
SCHEMBL9830028 0.87 KDM4E (0.41) KDM4EMAPTMEN1KMT2ARAB9A
SCHEMBL10470323 0.86 KDM4E (0.39) KDM4EMAPTMEN1KMT2ARAB9A
SCHEMBL9830269 0.78 KDM4E (0.45) KDM4EMAPTMEN1KMT2ARAB9A
SCHEMBL9831490 0.77 KDM4E (0.37) KDM4EMAPTMEN1KMT2ATSHR
SCHEMBL9831260 0.77 KDM4E (0.42) KDM4EMAPTMEN1KMT2ARAB9A
Hydrochloric Acid SCHEMBL10470525 0.77 KDM4E (0.36) KDM4EMAPTMEN1KMT2ATSHR
SCHEMBL9832126 0.77 KDM4E (0.47) KDM4EMAPTMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed