SCHEMBL9833006

SCHEMBL9833006

CN(C)c1ccc(NC(=O)C(C#N)C(=O)c2nn(-c3ccccc3)c3c2CSc2ccccc2-3)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 8/20 0.41
MAPT P10636 5/20 0.37
THRB P10828 1/20 0.37
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KMT2A Q03164 1/20 0.36
PIK3CD O00329 1/20 0.35
PIK3R2 O00459 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35
PIK3R5 Q8WYR1 1/20 0.35
PIK3R3 Q92569 1/20 0.35
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8111901 0.92 TP53 (0.42) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9833687 0.91 TP53 (0.41) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9316088 0.90 TP53 (0.44) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9832103 0.89 MAPT (0.43) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9833723 0.89 TP53 (0.41) TP53MAPTRAB9APIK3CDPIK3R2
SCHEMBL9832113 0.89 TP53 (0.40) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9831159 0.88 TP53 (0.40) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9831587 0.88 TP53 (0.40) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9316562 0.88 TP53 (0.46) TP53MAPTTHRBRAB9AL3MBTL1
SCHEMBL9833737 0.87 TP53 (0.45) TP53MAPTTHRBRAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed