SCHEMBL9833018

SCHEMBL9833018

Cc1ccccc1/C=C/c1cc2ccccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.51
CYP1A2 P05177 2/20 0.50
CYP2D6 P10635 2/20 0.50
MAPT P10636 2/20 0.50
NPSR1 Q6W5P4 2/20 0.50
BCHE P06276 1/20 0.50
ACHE P22303 1/20 0.50
IDO1 P14902 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
BRD4 O60885 1/20 0.46
ATP6V1B1 P15313 1/20 0.45
RAB9A P51151 4/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
THPO P40225 1/20 0.43
HIF1A Q16665 1/20 0.43
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
NPC1 O15118 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2458425 0.84 CYP2A6 (0.69) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL2458423 0.84 CYP2A6 (0.69) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL17433415 0.80 CYP2A6 (0.51) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL701421 0.80 CYP2A6 (0.51) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL701423 0.80 CYP2A6 (0.51) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL31448047 0.77 CYP2A6 (0.60) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL27764950 0.77 CYP2A6 (0.60) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL15359580 0.76 CYP2A6 (0.64) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL9834598 0.75 CYP2A6 (0.58) CYP2A6CYP1A2CYP2D6MAPTNPSR1
SCHEMBL538250 0.75 CYP2A6 (0.58) CYP2A6CYP1A2CYP2D6MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016004513-A1 ANTI-BACTERIAL PYRUVATE KINASE MODULATOR COMPOUNDS, COMPOSITIONS, USES AND METHODS SIMON FRASER UNIVERSITY (CA) 2016-01-14 WO disclosed
EP-0362695-B1 PYRROLOCARBAZOLE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS GÖDECKE AKTIENGESELLSCHAFT (DE) 1991-04-03 EP disclosed
US-4912107-A Pyrrolocarbazole derivatives, compositions containing them, and methods for using them GOEDECKE AKTIENGESELLSCHAFT (DE) 1990-03-27 US disclosed