SCHEMBL9836174

SCHEMBL9836174

O=C(O)C=Cc1cncc(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.48
RAB9A P51151 1/20 0.45
PADI4 Q9UM07 6/20 0.44
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC5 Q9UQL6 2/20 0.44
TNKS O95271 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
P4HTM Q9NXG6 1/20 0.42
KDM4E B2RXH2 4/20 0.42
HSD17B10 Q99714 3/20 0.42
CA12 O43570 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836170 1.00 HCAR2 (0.48) HCAR2RAB9APADI4HDAC3HDAC4
SCHEMBL30589032 0.84 HCAR2 (0.43) HCAR2RAB9APADI4HDAC1HDAC6
SCHEMBL3173354 0.80 PIK3C3 (0.49) HCAR2RAB9APADI4HDAC3HDAC4
SCHEMBL3173358 0.80 PIK3C3 (0.49) HCAR2RAB9APADI4HDAC3HDAC4
SCHEMBL17255822 0.80 KDM4E (0.50) HCAR2PADI4HDAC1HDAC6KDM4E
SCHEMBL17255821 0.80 KDM4E (0.50) HCAR2PADI4HDAC1HDAC6KDM4E
SCHEMBL6152906 0.79 CA12 (0.52) HCAR2RAB9AHDAC3HDAC4HDAC1
SCHEMBL6152908 0.79 CA12 (0.52) HCAR2RAB9AHDAC3HDAC4HDAC1
SCHEMBL1195656 0.78 BACE1 (0.53) HCAR2HDAC3HDAC4HDAC1HDAC7
SCHEMBL188332 0.78 BACE1 (0.53) HCAR2HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0210782-B1 PYRIDINE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Dainippon Pharmaceutical Co., Ltd. (JP) 1991-04-17 EP disclosed
US-4778796-A ω-(3-pyridyl)alkenamide derivatives and anti-allergenic pharmaceutical compositions containing same DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1988-10-18 US disclosed
EP-0210782-A2 Pyridine compounds, process for the preparation thereof and pharmaceutical composition containing the same Dainippon Pharmaceutical Co., Ltd. (JP) 1987-02-04 EP disclosed