SCHEMBL9836795

SCHEMBL9836795

Cc1cc(N=C=O)c(F)cc1Cl

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.42
TRPA1 O75762 1/20 0.42
TDP1 Q9NUW8 2/20 0.36
MAPK1 P28482 1/20 0.36
CD44 P16070 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7931545 0.84 TDP1 (0.45) CYP3A4TRPA1TDP1MAPK1ALDH1A1
SCHEMBL17310624 0.82 CYP3A4 (0.50) CYP3A4TRPA1TDP1MAPK1CD44
SCHEMBL10347965 0.82 TDP1 (0.39) CYP3A4TRPA1TDP1MAPK1ALDH1A1
SCHEMBL9837020 0.82 CYP3A4 (0.46) CYP3A4TRPA1TDP1ALDH1A1HPGD
SCHEMBL9730127 0.82 CYP3A4 (0.50) CYP3A4TRPA1TDP1MAPK1CD44
SCHEMBL17651437 0.81 CD44 (0.33) CD44ALDH1A1
SCHEMBL23240210 0.79 CYP3A4 (0.46) CYP3A4TRPA1TDP1MAPK1CD44
SCHEMBL29795916 0.79 CYP3A4 (0.50) CYP3A4TRPA1TDP1MAPK1CD44
SCHEMBL29795915 0.79 CYP3A4 (0.50) CYP3A4TRPA1TDP1MAPK1CD44
SCHEMBL23213379 0.79 CYP3A4 (0.50) CYP3A4TRPA1TDP1MAPK1CD44

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113248506-A Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-08-13 CN disclosed
CN-107001372-B Substituted aminopurine compounds, compositions thereof, and methods of treatment therewith 西格诺药品有限公司 2021-04-27 CN disclosed
EP-0241559-B1 OXAZOLIDINEDIONE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND HERBICIDES CONTAINING THE SAME SAGAMI CHEMICAL RESEARCH CENTER (JP) 1991-10-30 EP disclosed
US-4983751-A Chemical intermediates SAGAMI CHEMICAL RESEARCH CENTER (JP) 1991-01-08 US disclosed
US-4818272-A NONPHYTOTOXICITY FOR CROPS HELICAL STREAMS SAGAMI CHEMICAL RESEARCH CENTER (JP) 1989-04-04 US disclosed
EP-0241559-A1 OXAZOLIDINEDIONE DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND HERBICIDES CONTAINING THE SAME SAGAMI CHEMICAL RESEARCH CENTER (JP) 1987-10-21 EP disclosed