SCHEMBL9847015

SCHEMBL9847015

Nc1ccncc1C(N)Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 3/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
EPHX1 P07099 1/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1A2 P05177 2/20 0.41
TAAR1 Q96RJ0 2/20 0.40
MAOA P21397 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CYP2A6 P11509 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
AKT1 P31749 2/20 0.39
ANPEP P15144 1/20 0.38
HDAC8 Q9BY41 1/20 0.37
ROCK2 O75116 1/20 0.37
IKBKB O14920 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846958 0.83 IDO1 (0.43) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6
SCHEMBL7039235 0.78 CYP2D6 (0.41) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6
SCHEMBL7464343 0.78 EPHX1 (0.52) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6
SCHEMBL15972964 0.75 EPHX1 (0.41) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6
SCHEMBL9846993 0.74 KDM4E (0.44) ROCK2
SCHEMBL8867023 0.73 SLC6A2 (0.66) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6
SCHEMBL2477113 0.72 CYP2D6 (0.55) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6
SCHEMBL9041648 0.72 POLB (0.51) SIGMAR1CYP3A4CYP2C9CYP2C19AKT1
Hydrochloric Acid SCHEMBL9321422 0.72 SLC6A2 (0.63) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6
Hydrochloric Acid SCHEMBL6633931 0.71 CYP2D6 (0.54) SLC6A2SLC6A4SLC6A3EPHX1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0435222-A2 Aminopyridinylmethanols and aminomethylpyridinamines and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-07-03 EP disclosed