SCHEMBL9849174

SCHEMBL9849174

COC(=O)C1Cc2c(Br)cccc2CN1C(=O)OC

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.41
PTPN1 P18031 1/20 0.41
ABHD6 Q9BV23 3/20 0.40
AGTR2 P50052 2/20 0.39
PDE5A O76074 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16271276 1.00 CYP19A1 (0.41) CYP19A1PTPN1ABHD6AGTR2PDE5A
SCHEMBL29570670 1.00 CYP19A1 (0.41) CYP19A1PTPN1ABHD6AGTR2PDE5A
SCHEMBL31652041 1.00 CYP19A1 (0.41) CYP19A1PTPN1ABHD6AGTR2PDE5A
SCHEMBL32677218 0.90 CYP19A1 (0.45) CYP19A1PTPN1ABHD6AGTR2PDE5A
SCHEMBL32676636 0.90 CYP19A1 (0.45) CYP19A1PTPN1ABHD6AGTR2PDE5A
SCHEMBL16271289 0.90 PTPN1 (0.53) PTPN1ABHD6
SCHEMBL32676746 0.90 CYP19A1 (0.45) CYP19A1PTPN1ABHD6AGTR2PDE5A
SCHEMBL30069424 0.90 PTPN1 (0.53) PTPN1ABHD6
SCHEMBL20483181 0.90 PTPN1 (0.53) PTPN1ABHD6
SCHEMBL30069422 0.90 PTPN1 (0.53) PTPN1ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421436-A2 Substituted carboxytetrahydroisoquinolines and derivatives thereof having pharmaceutical activity WARNER-LAMBERT COMPANY (US) 1991-04-10 EP disclosed