SCHEMBL9849264

SCHEMBL9849264

CC(=O)NCCCCc1ccc(Br)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.59
KDM4E B2RXH2 2/20 0.54
F13A1 P00488 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPK1 P28482 1/20 0.50
HIF1A Q16665 1/20 0.50
PLAAT3 P53816 1/20 0.49
PLAAT5 Q96KN8 1/20 0.49
PLAAT2 Q9NWW9 1/20 0.49
PLAAT4 Q9UL19 1/20 0.49
GLA P06280 1/20 0.49
HPGD P15428 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
MTNR1A P48039 1/20 0.49
MTNR1B P49286 1/20 0.49
CNR1 P21554 1/20 0.48
CNR2 P34972 1/20 0.48
NLRP3 Q96P20 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL553085 0.87 KDM4E (0.70) KDM4EF13A1SMN1; SMN2HIF1APLAAT3
SCHEMBL5707308 0.84 KDM4E (0.77) KDM4EF13A1SMN1; SMN2MAPK1HIF1A
SCHEMBL425223 0.82 TRPV1 (0.65) HSP90AA1SMN1; SMN2KMT2AHPGDL3MBTL1
SCHEMBL16658733 0.81 TRPV1 (0.68) KDM4ESMN1; SMN2KMT2AMAPK1HIF1A
SCHEMBL16658698 0.81 TRPV1 (0.68) KDM4ESMN1; SMN2KMT2AMAPK1HIF1A
SCHEMBL16658696 0.81 TRPV1 (0.68) KDM4ESMN1; SMN2KMT2AMAPK1HIF1A
SCHEMBL16658695 0.81 TRPV1 (0.68) KDM4ESMN1; SMN2KMT2AMAPK1HIF1A
SCHEMBL5462618 0.81 TRPV1 (0.68) KDM4ESMN1; SMN2KMT2AMAPK1HIF1A
SCHEMBL16658697 0.81 TRPV1 (0.68) KDM4ESMN1; SMN2KMT2AMAPK1HIF1A
SCHEMBL5987763 0.79 KDM4E (0.58) KDM4EF13A1SMN1; SMN2KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421436-A2 Substituted carboxytetrahydroisoquinolines and derivatives thereof having pharmaceutical activity WARNER-LAMBERT COMPANY (US) 1991-04-10 EP disclosed