SCHEMBL9856196

SCHEMBL9856196

COc1ccc(C(=O)c2ccccc2)c(OCC(=O)O)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.76
KDM4E B2RXH2 1/20 0.70
LMNA P02545 4/20 0.62
HTT P42858 3/20 0.62
MAPK1 P28482 2/20 0.62
CYP1A2 P05177 2/20 0.62
CYP2C19 P33261 2/20 0.62
ALDH1A1 P00352 2/20 0.62
PGR P06401 1/20 0.62
CYP2D6 P10635 1/20 0.62
HPGD P15428 1/20 0.62
SLC6A2 P23975 1/20 0.62
PDE4A P27815 1/20 0.62
HRH1 P35367 1/20 0.62
SLC6A3 Q01959 1/20 0.62
PDE4D Q08499 1/20 0.62
NPC1 O15118 1/20 0.61
MAPT P10636 4/20 0.57
PTGDR2 Q9Y5Y4 2/20 0.57
SMN1; SMN2 Q16637 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9787076 0.90 POLB (0.74) POLBKDM4ELMNAHTTMAPK1
SCHEMBL9855260 0.90 PTGDR2 (0.68) POLBKDM4ELMNAHTTMAPK1
SCHEMBL16092725 0.90 MEN1 (0.61) POLBKDM4ELMNAHTTMAPK1
SCHEMBL11056067 0.88 POLB (0.71) POLBKDM4ELMNAHTTMAPK1
SCHEMBL21665232 0.87 NPC1 (0.73) POLBKDM4ELMNAHTTMAPK1
SCHEMBL16090169 0.87 POLB (0.63) POLBKDM4ELMNAMAPK1ALDH1A1
SCHEMBL3224251 0.86 NPC1 (0.81) POLBKDM4ELMNAHTTMAPK1
SCHEMBL30205105 0.86 NPC1 (0.81) POLBKDM4ELMNAHTTMAPK1
SCHEMBL1114933 0.85 POLB (0.64) POLBKDM4ELMNAHTTMAPK1
SCHEMBL29260273 0.84 POLB (0.67) POLBKDM4ELMNAHTTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0263492-B1 RETINOIDS, THEIR PREPARATION AND USE AS PHARMACEUTICAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 1991-03-13 EP disclosed
US-4900478-A SKIN DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-02-13 US disclosed
EP-0263492-A1 Retinoids, their preparation and use as pharmaceutical compounds F. HOFFMANN-LA ROCHE AG (CH) 1988-04-13 EP disclosed
US-4022908-A Use of certain 2-nitro-3-phenyl-alkoxybenzofurans in inhibiting growth of microorganisms and intermediates in the synthesis of said benzofurans RIKER LABORATORIES, INC. (US) 1977-05-10 US disclosed