SCHEMBL9857587

SCHEMBL9857587

O=C(O)c1c(OCc2ccccc2)cc(-c2ccccc2)cc1-c1ccc(F)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 7/20 0.51
RXRA P19793 1/20 0.50
RXRB P28702 1/20 0.50
RXRG P48443 1/20 0.50
MRGPRX4 Q96LA9 2/20 0.49
MCL1 Q07820 2/20 0.48
PTPN1 P18031 1/20 0.48
PTGER4 P35408 2/20 0.47
PTGER3 P43115 2/20 0.47
PTGER2 P43116 2/20 0.47
MGLL Q99685 1/20 0.46
MAP4K4 O95819 1/20 0.46
GPR34 Q9UPC5 1/20 0.46
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
DHODH Q02127 1/20 0.45
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
FOLH1 Q04609 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857813 0.77 DHODH (0.37) PTPN1MAP4K4DHODH
SCHEMBL9857652 0.76 PTPN1 (0.49) MCL1PTPN1MAP4K4DHODH
SCHEMBL2953824 0.75 MEN1 (0.49) PTGER1MCL1DHODH
SCHEMBL9857871 0.75 DHODH (0.50) PTPN1DHODHFOLH1
SCHEMBL9857473 0.74 DHODH (0.48) PTPN1MAP4K4MAPTDHODH
SCHEMBL31013973 0.73 PTGER1 (0.51) PTGER1MRGPRX4MCL1PTPN1LMNA
SCHEMBL6592997 0.73 MCL1 (0.51) PTGER1MRGPRX4MCL1PTPN1MAP4K4
SCHEMBL1316077 0.73 MCL1 (0.71) PTGER1MRGPRX4MCL1PTPN1PTGER4
SCHEMBL16624212 0.72 FFAR4 (0.62) PTGER1MCL1MGLLGPR34LMNA
SCHEMBL6245538 0.72 PTGER1 (0.65) PTGER1RXRARXRBRXRGMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072023-A Reacting lactone with ester anion to form cyclohexenone ester; oxidizing or dehydrogenating the intermediate E. R. SQUIBB & SONS, INC. (US) 1991-12-10 US disclosed
EP-0442495-A1 Process for preparing highly substituted phenyls E.R. SQUIBB & SONS, INC. (US) 1991-08-21 EP disclosed