SCHEMBL9861501

SCHEMBL9861501

Nc1ccc(N)c2c1C(=O)c1ccccc1C2(O)C(F)(F)C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 16/20 0.54
GRK6 P43250 1/20 0.48
CSNK1A1 P48729 2/20 0.44
CSNK1D P48730 2/20 0.44
CSNK1G1 Q9HCP0 2/20 0.44
ADORA2A P29274 2/20 0.44
FGR P09769 1/20 0.44
PIM1 P11309 1/20 0.44
MAOA P21397 1/20 0.44
DYRK1A Q13627 1/20 0.44
HIPK2 Q9H2X6 1/20 0.44
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
PABPC1 P11940 1/20 0.41
HPGD P15428 1/20 0.41
BLM P54132 1/20 0.41
KMT2A Q03164 1/20 0.41
MCL1 Q07820 1/20 0.41
PLEC Q15149 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861506 0.79 PDK2 (0.57) PDK2
SCHEMBL9861564 0.73 ADORA2A (0.36) PDK2GRK6CSNK1A1CSNK1DCSNK1G1
SCHEMBL9861335 0.73 PDK2 (0.48) PDK2MAOAMEN1HPGDKMT2A
SCHEMBL9861622 0.70 PDK2 (0.76) PDK2
SCHEMBL9861381 0.70 PDK2 (0.58) PDK2
SCHEMBL13128002 0.70 PDK2 (1.00) PDK2
SCHEMBL14907874 0.65 GRK6 (1.00) PDK2GRK6CSNK1A1CSNK1DCSNK1G1
SCHEMBL29361319 0.64 ADORA2A (1.00) GRK6CSNK1A1CSNK1DCSNK1G1ADORA2A
SCHEMBL525762 0.64 ADORA2A (1.00) GRK6CSNK1A1CSNK1DCSNK1G1ADORA2A
Hydrochloric Acid SCHEMBL8643536 0.62 ADORA2A (0.95) GRK6CSNK1A1CSNK1DCSNK1G1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008425-A Trifluoromethylation of carbonyl compounds ETHYL CORPORATION (US) 1991-04-16 US disclosed
US-4871877-A Gem-disubstituted cyclohexadienones and their production ETHYL CORPORATION (US) 1989-10-03 US disclosed