SCHEMBL9862189

SCHEMBL9862189

Clc1ccc(C2(Cn3ccnn3)CC(Br)CO2)c(Cl)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.67
CYP2C9 P11712 2/20 0.67
THRB P10828 1/20 0.37
CYP17A1 P05093 3/20 0.34
CYP21A2 P08686 3/20 0.34
CYP11B1 P15538 3/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
ADRA1A P35348 1/20 0.34
CCR1 P32246 5/20 0.33
CCR2 P41597 5/20 0.33
CCR4 P51679 4/20 0.33
CYP2C19 P33261 1/20 0.33
CYP19A1 P11511 4/20 0.33
CYP7A1 P22680 1/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21784834 0.86 CYP3A4 (0.46) CYP3A4CYP2C9THRBCYP17A1CYP21A2
Bromuconazole SCHEMBL22340 0.80 CYP3A4 (1.00) CYP3A4CYP2C9THRBLMNATSHR
Bromuconazole SCHEMBL3682832 0.80 CYP3A4 (1.00) CYP3A4CYP2C9THRBLMNATSHR
Bromuconazole SCHEMBL29360340 0.80 CYP3A4 (1.00) CYP3A4CYP2C9THRBLMNATSHR
SCHEMBL10574886 0.76 CYP3A4 (0.39) CYP3A4CYP2C9THRBUSP2ALDH1A1
Bromuconazole SCHEMBL1613562 0.76 CYP3A4 (0.89) CYP3A4CYP2C9THRBLMNATSHR
SCHEMBL4191977 0.76 CYP3A4 (0.43) CYP3A4CYP2C9THRBCYP17A1CYP21A2
Bromuconazole SCHEMBL28333287 0.75 CYP3A4 (0.87) CYP3A4CYP2C9THRBCYP17A1CYP21A2
SCHEMBL1279483 0.74 CYP3A4 (0.65) CYP3A4CYP2C9THRBCYP17A1CYP21A2
SCHEMBL9362816 0.74 CYP3A4 (0.38) CYP3A4CYP2C9THRBCYP17A1CYP21A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433194-A1 Fungicide composition with synergistic effect based on one morpholine and one triazole RHONE-POULENC AGROCHIMIE (FR) 1991-06-19 EP disclosed