SCHEMBL9862503

SCHEMBL9862503

CNC(=O)C(C)C(O)(Cn1cncn1)c1ccc(Cl)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 9/20 0.47
CYP2C9 P11712 7/20 0.47
CYP2C19 P33261 7/20 0.47
CYP1A2 P05177 5/20 0.47
CYP2D6 P10635 5/20 0.47
KCNH2 Q12809 2/20 0.47
LMNA P02545 3/20 0.43
MAPK1 P28482 2/20 0.43
CYP2B6 P20813 1/20 0.43
CYP3A5 P20815 1/20 0.43
CYP3A7 P24462 1/20 0.43
CYP3A43 Q9HB55 1/20 0.43
CYP46A1 Q9Y6A2 1/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 2/20 0.41
PKM P14618 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 2/20 0.39
HSP90AA1 P07900 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9862611 0.88 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
Water SCHEMBL9863844 0.86 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
Water SCHEMBL9863849 0.86 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL10924523 0.85 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9301060 0.85 CYP3A4 (0.47) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL10600188 0.83 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9663206 0.83 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9197506 0.83 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9523149 0.83 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6
SCHEMBL9197510 0.83 CYP3A4 (0.49) CYP3A4CYP2C9CYP2C19CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5047548-A 3-aryl-3-hydroxy-4-(1H-1,2,4-triazol-1-yl)butyramide and derivatives as antifungal agents PFIZER INC. (US) 1991-09-10 US disclosed
EP-0106515-B1 TRIAZOLE ANTI-FUNGAL AGENTS Pfizer Limited (GB) 1988-12-28 EP disclosed
US-4503063-A PLANTS AND ANIMALS PFIZER INC. (US) 1985-03-05 US disclosed
EP-0106515-A2 Triazole anti-fungal agents Pfizer Limited (GB) 1984-04-25 EP disclosed