SCHEMBL9867111

SCHEMBL9867111

COc1cc(NC(C)=O)c([N+](=O)[O-])cc1C(=O)NC1CCN(C/C=C/c2ccccc2)CC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 6/20 0.56
DRD4 P21917 8/20 0.52
DRD3 P35462 3/20 0.52
DRD2 P14416 2/20 0.52
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
LMNA P02545 2/20 0.47
MAPT P10636 1/20 0.47
CCR3 P51677 1/20 0.47
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
ADRA2A P08913 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
ACHE P22303 1/20 0.45
SLC6A2 P23975 1/20 0.45
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9867107 1.00 MCHR1 (0.56) MCHR1DRD4DRD3DRD2ALDH1A1
SCHEMBL9866636 0.88 MCHR1 (0.59) MCHR1DRD4DRD3DRD2ALDH1A1
SCHEMBL9866643 0.88 MCHR1 (0.59) MCHR1DRD4DRD3DRD2ALDH1A1
SCHEMBL9867273 0.86 DRD4 (0.65) MCHR1DRD4DRD3DRD2CYP1A2
Fumaric Acid SCHEMBL9866529 0.84 CYP3A4 (0.64) MCHR1DRD4DRD3DRD2CYP1A2
Fumaric Acid SCHEMBL9866524 0.84 CYP3A4 (0.64) MCHR1DRD4DRD3DRD2CYP1A2
SCHEMBL9866907 0.83 DRD4 (0.53) DRD4DRD3DRD2CYP1A2CYP3A4
Fumaric Acid SCHEMBL9867009 0.83 DRD4 (0.55) DRD4DRD3DRD2CYP1A2CYP3A4
Fumaric Acid SCHEMBL9867016 0.83 DRD4 (0.55) DRD4DRD3DRD2CYP1A2CYP3A4
SCHEMBL9867148 0.80 DRD4 (0.48) MCHR1DRD4DRD3DRD2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5026858-A Used for treating nausea, vomating, gastrointestinal disorders and centarl nervous system WALTON S.A. (ES) 1991-06-25 US disclosed