SCHEMBL9867694

SCHEMBL9867694

O=C(NC(=NCCCc1c[nH]cn1)NCCCSc1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 6/20 0.44
HRH4 Q9H3N8 4/20 0.44
KMT2A Q03164 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RECQL P46063 1/20 0.41
HRH1 P35367 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
POLB P06746 1/20 0.40
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HDAC1 Q13547 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HSP90AA1 P07900 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9866485 0.96 HRH4 (0.42) HRH2HRH4KMT2ANPC1RAB9A
SCHEMBL10369046 0.96 HRH4 (0.42) HRH2HRH4KMT2ANPC1RAB9A
SCHEMBL9866766 0.95 HRH2 (0.49) HRH2HRH4NPC1RAB9ASMN1; SMN2
SCHEMBL10369687 0.94 TDP1 (0.39) HRH2HRH4KMT2ANPC1RAB9A
SCHEMBL10369686 0.94 TDP1 (0.39) HRH2HRH4KMT2ANPC1RAB9A
SCHEMBL9865881 0.94 HPGD (0.46) HRH2HRH4KMT2ARAB9AHRH1
SCHEMBL9866763 0.94 NPC1 (0.42) HRH2HRH4KMT2ANPC1RAB9A
SCHEMBL9867435 0.94 NPC1 (0.42) HRH2HRH4KMT2ANPC1RAB9A
SCHEMBL9865867 0.90 HPGD (0.46) HRH2HRH4KMT2ANPC1RAB9A
SCHEMBL9865876 0.90 HPGD (0.46) HRH2HRH4KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021431-A H-1 antagonist, h-2 agonist for treating hypertension, cardiac disease or arterial occlusion HEUMANN PHARMA GMBH & CO. (DE) 1991-06-04 US disclosed