SCHEMBL9868972

SCHEMBL9868972

c1ccc2c(c1)CCN2C1=NCCN1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 1/20 0.47
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
TSHR P16473 2/20 0.41
CYP1A2 P05177 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HTT P42858 1/20 0.40
ALOX15 P16050 2/20 0.40
BRCA1 P38398 1/20 0.40
SRD5A1 P18405 1/20 0.40
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2123689 0.74 ROCK1 (0.49) ROCK1LMNATP53MAPK1SMN1; SMN2
SCHEMBL11883161 0.74 EED (0.46) TSHRCYP1A2
SCHEMBL9562173 0.71 TP53 (0.44) ROCK1LMNATP53MAPK1SMN1; SMN2
SCHEMBL10620614 0.71 MEN1 (0.51) LMNACYP1A2ALDH1A1ALOX15MEN1
SCHEMBL3239758 0.70 ROCK1 (0.61) ROCK1LMNATP53MAPK1SMN1; SMN2
SCHEMBL29721693 0.70 ROCK1 (0.61) ROCK1LMNATP53MAPK1SMN1; SMN2
Hydrochloric Acid SCHEMBL8675065 0.69 CYP1A2 (0.65) TSHRCYP1A2ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL27693256 0.69 ROCK1 (0.59) ROCK1LMNATP53MAPK1SMN1; SMN2
SCHEMBL6071629 0.68 ROCK1 (0.62) ROCK1LMNATP53MAPK1SMN1; SMN2
SCHEMBL29721478 0.68 ROCK1 (0.62) ROCK1LMNATP53MAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3935199-A ANALEPTIC MEAD JOHNSON & COMPANY (US) 1976-01-27 US claimed
US-5017584-A Antidepressant 2-(4,5-dihydro-1H-imidazolyl)-dihydro-1H-indoles, -1,2,3,4-tetrahydroquinolines and -1H-indoles, and methods of use thereas STERLING DRUG INC. (US) 1991-05-21 US disclosed