SCHEMBL9869637

SCHEMBL9869637

COc1ccc(-c2c(S)ncc(C)c2C#N)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 4/20 0.44
KDM4E B2RXH2 6/20 0.44
ALDH1A1 P00352 5/20 0.44
GAA P10253 2/20 0.44
PTPN1 P18031 2/20 0.43
NPSR1 Q6W5P4 5/20 0.43
RXFP1 Q9HBX9 5/20 0.43
PPARG P37231 1/20 0.43
HTT P42858 1/20 0.43
NCOA2 Q15596 1/20 0.43
NCOA1 Q15788 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
NTRK1 P04629 1/20 0.42
PIM1 P11309 1/20 0.42
POLB P06746 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
MAPT P10636 6/20 0.41
MEN1 O00255 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL245539 0.80 ADORA1 (0.46) ADORA1KDM4EALDH1A1GAAPTPN1
SCHEMBL3359383 0.71 KDM4E (0.60) ADORA1KDM4EALDH1A1GAAPTPN1
SCHEMBL16294362 0.69 KDM4E (0.70) KDM4EALDH1A1GAANPSR1RXFP1
SCHEMBL8473714 0.68 KDM4E (0.50) ADORA1KDM4EALDH1A1GAAPTPN1
SCHEMBL23957342 0.67 PTPN1 (0.50) ADORA1KDM4EALDH1A1GAAPTPN1
SCHEMBL28185544 0.67 CYP11B1 (0.54) ADORA1KDM4EALDH1A1GAAPTPN1
SCHEMBL23629573 0.67 PTPN1 (0.50) ADORA1KDM4EALDH1A1GAAPTPN1
SCHEMBL29152123 0.66 PTPN1 (0.51) ADORA1KDM4EALDH1A1GAAPTPN1
SCHEMBL12874583 0.66 KDM4E (0.63) ADORA1KDM4EALDH1A1GAANPSR1
SCHEMBL15712825 0.66 PTPN1 (0.56) ADORA1KDM4EALDH1A1GAAPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006532-A Enzyme inhibitor; antiinflammatory agents MERCK & CO. INC., INC. (US) 1991-04-09 US disclosed