SCHEMBL9870175

SCHEMBL9870175

COC1=C(C(=O)OCc2ccccc2)N2C(=O)CC2C1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ELANE P08246 9/20 0.58
GPBAR1 Q8TDU6 3/20 0.43
ALDH1A1 P00352 1/20 0.43
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870539 0.88 ELANE (0.56) ELANEGPBAR1ALDH1A1SLC6A2SLC6A3
SCHEMBL11175452 0.86 ELANE (0.54) ELANEGPBAR1ALDH1A1SLC6A2SLC6A3
SCHEMBL11231753 0.82 ELANE (0.57) ELANEGPBAR1ALDH1A1SLC6A2SLC6A3
SCHEMBL9870437 0.82 ELANE (0.57) ELANEGPBAR1SLC6A2SLC6A3KMT2A
SCHEMBL10570187 0.81 ELANE (0.51) ELANEGPBAR1
SCHEMBL9870805 0.79 ELANE (0.48) ELANEGPBAR1
SCHEMBL10570612 0.79 ELANE (0.56) ELANEGPBAR1SLC6A2SLC6A3KMT2A
SCHEMBL11110289 0.78 ELANE (0.53) ELANEGPBAR1
SCHEMBL9870806 0.78 ELANE (0.52) ELANEGPBAR1ALDH1A1SLC6A2SLC6A3
SCHEMBL11115998 0.78 ELANE (0.52) ELANEGPBAR1SLC6A2SLC6A3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5021566-A Carbapenicillins; preservatives; antiseptics; grampositive and gram negative bacteria MERCK & CO. INC. (US) 1991-06-04 US disclosed
US-4820817-A Process for preparing 3-substituted-6-substituted-7-oxo-1-azabicycl(3.2.0)-hept-2-ene-2-carboxylic acid MERCK & CO., INC. (US) 1989-04-11 US disclosed
US-4745188-A ANTIBIOTICS, SULFIDING MERCK & CO., INC. (US) 1988-05-17 US disclosed
US-4707547-A AMINATION TO FORM ANTIBIOTIC MERCK & CO., INC. (US) 1987-11-17 US disclosed
US-4530841-A Antibiotic containing hetero ring MERCK & CO., INC. (US) 1985-07-23 US disclosed
EP-0134301-A1 6-(1'-Hydroxyethyl)-3-substituted amino-1-azabicyclo(3.2.0)-hept-2-en-7-one-2-carboxylic acid MERCK & CO. INC. (US) 1985-03-20 EP disclosed
US-4369187-A AMINO ACID DERIVATIVE ANTIBIOTICS MERCK & CO., INC. (US) 1983-01-18 US disclosed
US-4357342-A 1-Azabicyclo[3.2.0]heptan-3,7-dione-2-carboxylic acid MERCK & CO., INC. (US) 1982-11-02 US disclosed
US-4318912-A 6-(1-Hydroxyethyl)-3-substituted-1-azabicyclo(3.2.0)-hept-2-en-7-one-2-carboxylic acid MERCK & CO., INC. (US) 1982-03-09 US disclosed