SCHEMBL9870644

SCHEMBL9870644

CC(C)c1nc(C(C)C)c(C(=O)O)c(-c2ccc(F)cc2)c1CC=CO

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GCGR P47871 18/20 0.56
DPP4 P27487 1/20 0.43
DPP8 Q6V1X1 1/20 0.43
DPP9 Q86TI2 1/20 0.43
ESR1 P03372 1/20 0.42
HMGCR P04035 1/20 0.42
CHRM1 P11229 1/20 0.42
TBXA2R P21731 1/20 0.42
PDE4A P27815 1/20 0.42
ADRA1A P35348 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9870949 1.00 GCGR (0.56) GCGRDPP4DPP8DPP9ESR1
SCHEMBL9871037 0.84 GCGR (0.52) GCGR
SCHEMBL9871041 0.84 GCGR (0.52) GCGR
SCHEMBL2651071 0.82 GCGR (0.56) GCGRDPP4DPP8DPP9
SCHEMBL2647594 0.80 GCGR (0.70) GCGR
SCHEMBL2646545 0.76 GCGR (0.77) GCGRESR1HMGCRCHRM1TBXA2R
SCHEMBL5098308 0.76 GCGR (0.50) GCGRDPP4DPP8DPP9
SCHEMBL8879628 0.75 DHODH (0.55) GCGRDPP4DPP8DPP9
SCHEMBL27293870 0.75 GCGR (0.49) GCGRDPP4DPP8DPP9
SCHEMBL9870958 0.74 GCGR (0.72) GCGRDPP4DPP8DPP9ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed