SCHEMBL9871355

SCHEMBL9871355

CCc1cc(-c2ccc(F)cc2)c(/C=C/[C@H](O)C[C@H](O)CC(=O)O)c(CC)n1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 10/20 0.51
NR1I2 O75469 2/20 0.51
PDE4D Q08499 2/20 0.51
NR4A2 P43354 1/20 0.51
ESR1 P03372 1/20 0.51
CHRM1 P11229 1/20 0.51
TBXA2R P21731 1/20 0.51
PDE4A P27815 1/20 0.51
ADRA1A P35348 1/20 0.51
ALDH1A1 P00352 1/20 0.50
CYP3A4 P08684 1/20 0.50
PDE6D O43924 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871365 1.00 HMGCR (0.51) HMGCRNR1I2PDE4DNR4A2ESR1
SCHEMBL9871004 0.82 HMGCR (0.55) HMGCRNR1I2PDE4DNR4A2ESR1
SCHEMBL9022660 0.82 HMGCR (0.55) HMGCRNR1I2PDE4DNR4A2ESR1
SCHEMBL9872409 0.82 HMGCR (0.60) HMGCRNR1I2PDE4DNR4A2ESR1
SCHEMBL9872399 0.82 HMGCR (0.60) HMGCRNR1I2PDE4DNR4A2ESR1
SCHEMBL10424094 0.81 HMGCR (0.54) HMGCRNR1I2PDE4DNR4A2ESR1
SCHEMBL10424098 0.81 HMGCR (0.54) HMGCRNR1I2PDE4DNR4A2ESR1
SCHEMBL9871185 0.79 HMGCR (0.64) HMGCRNR1I2PDE4DESR1CHRM1
SCHEMBL9871701 0.78 HMGCR (0.63) HMGCRNR1I2PDE4DESR1CHRM1
SCHEMBL9871697 0.78 HMGCR (0.63) HMGCRNR1I2PDE4DESR1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US claimed
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed