SCHEMBL9879875

SCHEMBL9879875

CCCCCCCCCCCCC(CC(=O)c1ccc(NCc2ccc3ccc4nc(C)[nH]c(=O)c4c3c2)cc1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TYMS P04818 12/20 0.54
FPGS Q05932 1/20 0.42
PPARG P37231 1/20 0.40
PPARD Q03181 1/20 0.40
PPARA Q07869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447643 0.90 TYMS (0.56) TYMSFPGS
SCHEMBL6446417 0.90 TYMS (0.64) TYMS
SCHEMBL6446398 0.90 TYMS (0.64) TYMS
SCHEMBL9422204 0.86 TYMS (0.57) TYMS
SCHEMBL6651090 0.82 TYMS (0.48) TYMSFPGS
SCHEMBL6648735 0.82 TYMS (0.58) TYMS
SCHEMBL6447490 0.81 TYMS (0.61) TYMS
SCHEMBL6842975 0.79 TYMS (0.53) TYMS
SCHEMBL6447640 0.78 TYMS (0.52) TYMS
SCHEMBL9422199 0.77 TYMS (0.55) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019700-A1 PHARMACEUTICALLY ACTIVE BENZOQUINAZOLINE COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-26 WO disclosed